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Search Results

Showing results 21 to 40 of 62.

Article

Validation of a high-throughput calcium mobilization assay for the human trace amine-associated receptor 1

January 01, 2021
Article

Design, synthesis, and structure-activity relationship studies of (4-alkoxyphenyl)glycinamides and bioisosteric 1,3,4-oxadiazoles as GPR88 agonists

December 10, 2020
Article

Synthesis and pharmacological evaluation of 1-phenyl-3-thiophenylurea derivatives as cannabinoid type-1 receptor allosteric modulators

November 14, 2019
Article

Functionalized 6-(piperidin-1-yl)-8,9-diphenyl purines as peripherally restricted inverse agonists of the CB1 receptor

July 11, 2019
Article

The dopamine, serotonin and norepinephrine releasing activities of a series of methcathinone analogs in male rat brain synaptosomes

March 01, 2019
Article

Diarylureas containing 5-membered heterocycles as cb1 receptor allosteric modulators: Design, synthesis, and pharmacological evaluation

January 16, 2019
Article

Comparative neuropharmacology of N-(2-methoxybenzyl)-2,5-dimethoxyphenethylamine (NBOMe) hallucinogens and their 2C counterparts in male rats

November 01, 2018
Article

Potent and selective tetrahydroisoquinoline kappa opioid receptor antagonists of lead compound (3 R)- N-[1 R)-1-(Cyclohexylmethyl)-2-methylpropyl]-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (CDTic)

September 13, 2018
Article

Potent and selective tetrahydroisoquinoline kappa opioid receptor antagonists of lead compound (3r)-7-hydroxy-n-[(1s)-2-methyl-1-(piperidin-1-ylmethyl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (pdtic)

September 13, 2018
Article

Development of serotonin transporter reuptake inhibition assays using JAR cells

September 01, 2018
Article

Discovery of a potent, selective, and brain-penetrant small molecule that activates the orphan receptor GPR88 and reduces alcohol intake

August 09, 2018
Article

Fluorinated phenmetrazine "legal highs" act as substrates for high-affinity monoamine transporters of the SLC6 family

May 15, 2018
Article

Development of norepinephrine transporter reuptake inhibition assays using SK-N-BE(2)C cells

May 01, 2018
Article

Synthesis and evaluation of orexin-1 receptor antagonists with improved solubility and CNS permeability

March 21, 2018
Article

Discovery of novel proline-based neuropeptide FF receptor antagonists

October 18, 2017
Article

Novel diarylurea based allosteric modulators of the cannabinoid CB1 receptor: Evaluation of importance of 6-pyrrolidinylpyridinyl substitution

September 14, 2017
Article

Simple tetrahydroisoquinolines are potent and selective kappa opioid receptor antagonists

July 13, 2017
Patent

Phenylmorpholines and Analogues Thereof

April 11, 2017
Article

Development and validation of a high-throughput calcium mobilization assay for the orphan receptor GPR88

March 27, 2017
Article

Design, synthesis and pharmacological evaluation of 4-hydroxyphenylglycine and 4-hydroxyphenylglycinol derivatives as GPR88 agonists

January 15, 2017