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Showing results 1 to 20 of 130.
Article
A highly G protein-biased mu opioid receptor agonist, sr-17018, has low in vivo efficacy in primates
July 01, 2024
Article
Dopamine D1 receptor in medial prefrontal cortex mediates the effects of TAAR1 activation on chronic stress-induced cognitive and social deficits
July 01, 2024
Article
TAAR1 in dentate gyrus is involved in chronic stress-induced impairments in hippocampal plasticity and cognitive function
June 08, 2024
Article
The imidazoline I2 receptor agonist 2-BFI reduces abuse-related effects of morphine: Self-administration and drug discrimination
March 01, 2024
Article
Effects of a highly G Protein-Biased Mu Opioid Receptor Agonist, SR-17018, in Non-human Primates
June 01, 2023
Article
Isoquinolone derivatives as lysophosphatidic acid receptor 5 (LPA5) antagonists: Investigation of structure-activity relationships, ADME properties and analgesic effects
December 05, 2022
Patent
Proline-based neuropeptide FF receptor modulators
November 08, 2022
Article
Selective TAAR1 agonists induce conditioned taste aversion
October 01, 2022
Article
In vitro and in vivo pharmacology of nine novel synthetic cannabinoid receptor agonists
October 01, 2022
Article
TAAR1 regulates drug-induced reinstatement of cocaine-seeking via negatively modulating CaMKIIα activity in the NAc
April 01, 2022
Article
Neuropeptide B/W receptor 1 peptidomimetic agonists: Structure-activity relationships and plasma stability
March 05, 2022
Article
RTICBM-74 Is a brain-penetrant cannabinoid receptor subtype 1 allosteric modulator that reduces alcohol intake in rats
March 01, 2022
Article
Exploring determinants of agonist efficacy at the CB1 cannabinoid receptor: Analogues of the synthetic cannabinoid receptor agonist EG-018
February 01, 2022
Article
Development of 3-(4-chlorophenyl)-1-(phenethyl)urea analogues as allosteric modulators of the cannabinoid type-1 receptor: RTICBM-189 is brain penetrant and attenuates reinstatement of cocaine-seeking behavior
January 13, 2022
Article
Activation of trace amine-associated receptor 1 attenuates nicotine withdrawal-related effects
January 01, 2022
Article
The selective TAAR1 partial agonist RO5263397 promoted novelty recognition memory in mice
November 01, 2021
Article
Identification of a novel neuropeptide S receptor antagonist scaffold based on the SHA-68 core
October 06, 2021
Patent
Diarylureas as CB1 allosteric modulators
August 10, 2021
Article
Age-specific treatment effects of orexin/hypocretin-receptor antagonism on methamphetamine-seeking behavior
July 01, 2021
Article
Rational design of cannabinoid type-1 receptor allosteric modulators: Org27569 and PSNCBAM-1 hybrids
July 01, 2021