Search Results
Showing results 1 to 20 of 69.
Patent
Heterocyclic apelin receptor (APJ) agonists and uses thereof
March 12, 2024
Article
Discovery of 1,3-disubstituted pyrazole peripheral cannabinoid receptor partial agonists
September 01, 2023
Patent
Apelin receptor (APJ) agonists and uses thereof
August 01, 2023
Article
The monoacylglycerol lipase inhibitor ABX-1431 does not improve alcoholic liver disease
May 29, 2023
Article
Improvement of the metabolic stability of GPR88 agonist RTI-13951-33: Design, synthesis, and biological evaluation
February 23, 2023
Patent
Apelin receptor (APJ) agonists and uses thereof
December 27, 2022
Chapter
Recent advances in the development of small-molecule apelin receptor agonists for cardiovascular and metabolic diseases
December 21, 2022
Article
Structure-activity relationship development efforts towards peripherally selective analogs of the cannabinoid receptor partial agonist BAY 59-3074
September 02, 2022
Patent
Apelin receptor (APJ) agonists and uses thereof
August 02, 2022
Article
Synthesis and characterization of an orally bioavailable small molecule agonist of the apelin receptor
July 15, 2022
Article
Evaluation of amide bioisosteres leading to 1,2,3-triazole containing compounds as GPR88 agonists: Design, synthesis, and structure-activity relationship studies
August 26, 2021
Article
"Photo-Rimonabant": Synthesis and biological evaluation of novel photoswitchable molecules derived from Rimonabant lead to a highly selective and nanomolar "Cis-On" CB1R antagonist
May 05, 2021
Article
Peripherally selective CB1 receptor antagonist improves symptoms of metabolic syndrome in mice
April 09, 2021
Article
Pyrazole agonist of the apelin receptor improves symptoms of metabolic syndrome in mice
March 25, 2021
Patent
Apelin receptor (APJ) agonists and uses thereof
March 23, 2021
Article
Aplnr knockout mice display sex-specific changes in conditioned fear
February 26, 2021
Article
Design, synthesis, and structure-activity relationship studies of (4-alkoxyphenyl)glycinamides and bioisosteric 1,3,4-oxadiazoles as GPR88 agonists
December 10, 2020
Article
Behavioral assessment of rimonabant under acute and chronic conditions
July 15, 2020
Patent
Diaryl purine derivatives with improved bioavailability
June 30, 2020
Article
Identification of potent pyrazole based APELIN receptor (APJ) agonists
February 15, 2020