David Hesk

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Synthesis and pharmacological validation of a novel radioligand for the orphan GPR88 receptor

Identification of a potent human trace amine-associated receptor 1 antagonist

Metallaphotoredox aryl and alkyl radiomethylation for PET ligand discovery

New methodologies for labelling with hydrogen isotopes

Hydrogen isotope exchange labelling: A brief update

Base metal-catalyzed hydrogen isotope exchange

Synthesis of [H-3] and [C-14]genipin

Highlights of C (sp2 )-H hydrogen isotope exchange reactions

Deuterated active pharmaceutical ingredients: A science based proposal for synthesis, analysis, and control. Part 1: Framing the problem

Iridium-catalysed hydrogen isotope exchange of amino acid and peptide molecules

Ni(I)-X Complexes Bearing a Bulky α-Diimine Ligand: Synthesis, structure, and superior catalytic performance in the hydrogen isotope exchange in pharmaceuticals

Site-selective nickel-catalyzed hydrogen isotope exchange in h-heterocycles and its application to the tritiation of pharmaceuticals

Synthesis of 3 H, 13 C 2 , 2 H 4 14 C-SCH 430765 and 35 S-SCH 500946, potent and selective inhibitors of the NPY 5 receptor.

Synthesis of 3H, 13C2, 2H414C‐SCH 430765 and 35S‐SCH 500946, potent and selective inhibitors of the NPY5 receptor

S-34: A new opportunity for the efficient synthesis of stable isotope labeled compounds

34S: A new opportunity for the efficient synthesis of stable isotope labeled compounds

A general strategy for site-selective incorporation of deuterium and tritium into pyridines, diazines, and pharmaceuticals

Photoredox-catalyzed deuteration and tritiation of pharmaceutical compounds

Palladium mediated C-H tritiation

Electrochemical bromination of late stage intermediates and drug molecules